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PMID: 12746500 Published · ppublish English Journal Article

Specificity of short interfering RNA determined through gene expression signatures.

Semizarov D, Frost L, Sarthy A, Kroeger P, Halbert DN, Fesik SW

Abstract

Short interfering RNA (siRNA) is widely used for studying gene function and holds great promise as a tool for validating drug targets and treating disease. A critical assumption in these applications is that the effect of siRNA on cells is specific, i.e., limited to the specific knockdown of the target gene. In this article, we characterize the specificity of siRNA by applying gene expression profiling. Several siRNAs were designed against different regions of the same target gene for three different targets. Their effects on cells were compared by using DNA microarrays to generate gene expression signatures. When the siRNA design and transfection conditions were optimized, the signatures for different siRNAs against the same target were shown to correlate very closely, whereas the signatures for different genes revealed no correlation. These results indicate that siRNA is a highly specific tool for targeted gene knockdown, establishing siRNA-mediated gene silencing as a reliable approach for large-scale screening of gene function and drug target validation.

MeSH Terms
Gene Expression Oligonucleotide Array Sequence Analysis RNA, Small Interfering/metabolism Reverse Transcriptase Polymerase Chain Reaction
Chemicals
RNA, Small Interfering
Authors & Affiliations
6 authors, click to expand affiliations / ORCID
Semizarov Dimitri
Global Pharmaceutical Research and Development, Abbott Laboratories, 100 Abbott Park Road, IL 60064, USA. [email protected]
Frost Leigh
Sarthy Aparna
Kroeger Paul
Halbert Donald N
Fesik Stephen W
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Article Info
Journal
Proceedings of the National Academy of Sciences of the United States of America
Abbr.
Proc Natl Acad Sci U S A
ISSN
0027-8424
Published
2003-05-27
Epub
2003-00-13
Pages
6347-52
Language
English
Region
United States
NLM ID
7505876
PMCID
PMC164449
Subset
IM
Corrections
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