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PMID: 15134285 Published · ppublish English Journal Article Review

Rimonabant Sanofi-Synthélabo.

Current opinion in investigational drugs (London, England : 2000) ·Vol. 5 ·No. 4 ·2004-04-00 ·Pages 430-5

Fernandez JR, Allison DB

Abstract

Rimonabant, an antagonist of central cannabinoid type 1 (CB1) receptors, is being developed by Sanofi-Synthélabo for the potential treatment of obesity and as a potential smoking cessation agent. Phase III trials were initiated for obesity in August 2001 and were ongoing in September 2003. By September 2002, the compound had entered phase III trials for smoking cessation, and these trials were ongoing in September 2003.

MeSH Terms
Animals Anti-Obesity Agents/chemical synthesis,chemistry,pharmacokinetics Antipsychotic Agents/chemical synthesis,chemistry,pharmacokinetics Appetite Depressants/chemical synthesis,chemistry,pharmacokinetics Clinical Trials as Topic Humans Obesity/drug therapy Piperidines/chemical synthesis,chemistry,pharmacokinetics Potassium Channel Blockers/chemical synthesis,chemistry,pharmacokinetics Pyrazoles/chemical synthesis,chemistry,pharmacokinetics Receptor, Cannabinoid, CB1/antagonists & inhibitors Rimonabant Smoking Cessation Structure-Activity Relationship
Chemicals
Anti-Obesity Agents Antipsychotic Agents Appetite Depressants Piperidines Potassium Channel Blockers Pyrazoles Receptor, Cannabinoid, CB1 Rimonabant
Authors & Affiliations
2 authors, click to expand affiliations / ORCID
Fernandez Jose R
University of Alabama at Birmingham, Department of Nutrition Sciences, Ryals Public Health Building, 1665 University Blvd, Birmingham, AL 35294-0022, USA.
Allison David B
Article Info
Journal
Current opinion in investigational drugs (London, England : 2000)
Abbr.
Curr Opin Investig Drugs
ISSN
1472-4472
Published
2004-04-00
Pages
430-5
Language
English
Region
England
NLM ID
100965718
Subset
IM
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