Abstract
The efficacy of various drugs used to treat ulcerative colitis, (sulfasalazine, 5-aminosalicylate, hydrocortisone) was investigated in a model of acetic acid-induced colitis in the rat. Subsequently, we tested the ability of antioxidant/5-lipoxygenase inhibitors (gossypol and nordihydroguiaretic acid [NDGA]) and a cyclooxygenase inhibitor (indomethacin) to attenuate the macroscopic colonic damage and/or neutrophil influx (myeloperoxidase activity [MPO]) associated with this model of colitis. Oral pretreatment with either sulfasalazine, gossypol, or NDGA significantly decreased colonic MPO activity induced by acetic acid. Intrarectal administration of such drugs resulted in an even larger reduction of the colonic inflammation, with gossypol being the most potent compound. Oral or intrarectal administration of corticosteroids (dexamethasone, hydrocortisone) also attenuated the parameters of acetic acid induced colitis. In contrast, pretreatment with indomethacin was ineffective, or when administered daily after colitis induction, indomethacin actually increased colonic neutrophil influx significantly. Our data suggest that both the route of drug administration and dosing regimen employed affect the antiinflammatory potency and/or efficacy of compounds on colitis induced by acetic acid in the rat. Drugs which were effective against this colitis may act by scavenging of oxygen derived free radicals.
MeSH Terms
Acetates
Acetic Acid
Aminosalicylic Acids/therapeutic use
Animals
Anti-Inflammatory Agents
Colitis, Ulcerative/chemically induced,drug therapy
Dexamethasone/therapeutic use
Disease Models, Animal
Gossypol/therapeutic use
Hydrocortisone/therapeutic use
Indomethacin/therapeutic use
Intestinal Mucosa/drug effects,pathology
Leukocyte Count
Male
Masoprocol/therapeutic use
Mesalamine
Neutrophils/enzymology
Peroxidase/metabolism
Rats
Rats, Inbred Strains
Sulfasalazine/therapeutic use
Chemicals
Acetates
Aminosalicylic Acids
Anti-Inflammatory Agents
Sulfasalazine
Mesalamine
Masoprocol
Dexamethasone
Peroxidase
Gossypol
Acetic Acid
Hydrocortisone
Indomethacin
Authors & Affiliations
5 authors, click to expand affiliations / ORCID
Fitzpatrick L R
Gastrointestinal Pharmacology Department, Rorer Central Research, Horsham, PA 19044.
Bostwick J S
Renzetti M
Pendleton R G
Decktor D L
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