Abstract
Jasplakinolide is a cyclodepsipeptide which represents a new class of antifungal agents with potent activity against Candida albicans. Jasplakinolide is fungicidal against C. albicans with both a MIC and a minimum lethal concentration of 25 micrograms/ml in a broth dilution assay. This activity compares to that of the imidazole miconazole nitrate, which had a MIC of 6.2 micrograms/ml and a minimum lethal concentration of 50 micrograms/ml in the same assay. Topical administration of 2% jasplakinolide cream against a murine vaginal C. albicans infection was equivalent in efficacy to administration of miconazole nitrate at 2%. Subcutaneous administration of jasplakinolide was not effective against a systemic murine C. albicans infection.
MeSH Terms
Animals
Antifungal Agents/metabolism,pharmacology,therapeutic use,toxicity
Candida/drug effects,metabolism
Candidiasis/drug therapy
Candidiasis, Vulvovaginal/drug therapy
Chemical Phenomena
Chemistry
Depsipeptides
Female
Mice
Mice, Inbred ICR
Microbial Sensitivity Tests
Peptides, Cyclic/metabolism,pharmacology,therapeutic use,toxicity
Chemicals
Antifungal Agents
Depsipeptides
Peptides, Cyclic
jasplakinolide
Authors & Affiliations
3 authors, click to expand affiliations / ORCID
Scott V R
Department of Antimicrobial Chemotherapy, Syntex Research, Palo Alto, California 94304.
Boehme R
Matthews T R
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