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PMID: 4313200 Published · ppublish English Journal Article

Inhibition of hormone-sensitive adenyl cyclase by phenothiazines.

Wolff J, Jones AB

Abstract

Chlorpromazine (3 x 10(-4)M) prevents the stimulation of adenyl cyclase activity in thyroid membranes produced by thyrotropin and prostaglandin, ACTH stimulation of adenyl cyclase in adrenal tissue, and glucagon- and epinephrine-stimulation of adenyl cyclase activity in liver. Baseline activity is unaffected. Parathyroid hormone stimulation of kidney preparations was not inhibited under these conditions. At chlorpromazine concentrations >3 x 10(-4)M F(-)-stimulated cyclase activity of thyroid and adrenal tissue was increased. Other phenothiazines, trifluoperazine, and prochlorperazine, have similar effects on thyrotropin and F(-)-stimulated cyclase activity of thyroid. Na(+)- K(+)-dependent ATPase of thyroid is also inhibited by chlorpromazine. Since thymol causes a similar dissociation of hormone- and F(-)-stimulated adenyl cyclase, it is concluded that the surface properties of these agents best account for their effects on adenyl cyclase.

MeSH Terms
Adenine Nucleotides Adenylyl Cyclase Inhibitors Adrenal Glands/enzymology Adrenocorticotropic Hormone/antagonists & inhibitors Animals Cattle Cell Membrane/enzymology Chlorpromazine/pharmacology Enzyme Inhibitors Epinephrine/antagonists & inhibitors Fluorides/pharmacology Glucagon/antagonists & inhibitors Kidney/enzymology Liver/enzymology Phenothiazines/pharmacology Pituitary Hormones, Anterior/antagonists & inhibitors Prochlorperazine/pharmacology Prostaglandin Antagonists Stimulation, Chemical Thymol/pharmacology Thyroid Gland/cytology,enzymology Thyrotropin/antagonists & inhibitors Trifluoperazine/pharmacology
Chemicals
Adenine Nucleotides Adenylyl Cyclase Inhibitors Enzyme Inhibitors Phenothiazines Pituitary Hormones, Anterior Prostaglandin Antagonists Trifluoperazine Thymol Adrenocorticotropic Hormone Thyrotropin Glucagon Fluorides Chlorpromazine Prochlorperazine Epinephrine
Authors & Affiliations
2 authors, click to expand affiliations / ORCID
Wolff J
Jones A B
References (15)
15 references, click to expand
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Article Info
Journal
Proceedings of the National Academy of Sciences of the United States of America
Abbr.
Proc Natl Acad Sci U S A
ISSN
0027-8424
Published
1970-02-00
Pages
454-9
Language
English
Region
United States
NLM ID
7505876
PMCID
PMC282924
Subset
IM
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