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PMID: 9779453 Published · ppublish English Journal Article Research Support, Non-U.S. Gov't Research Support, U.S. Gov't, P.H.S.

Inhibition of [3H]dopamine translocation and [3H]cocaine analog binding: a potential screening device for cocaine antagonists.

Methods in enzymology ·Vol. 296 ·1998-00-00 ·Pages 248-59

Reith ME, Xu C, Carroll FI, Chen NH

Abstract

暂无摘要

MeSH Terms
Animals Biological Transport Carrier Proteins/metabolism Cell Fractionation/methods Cell Membrane/metabolism,ultrastructure Cocaine/analogs & derivatives,antagonists & inhibitors,pharmacokinetics Corpus Striatum/metabolism Dopamine/metabolism Dopamine Plasma Membrane Transport Proteins Drug Design Membrane Glycoproteins Membrane Transport Proteins Nerve Tissue Proteins Radioligand Assay/methods Rats Sodium/metabolism Software Tritium
Chemicals
Carrier Proteins Dopamine Plasma Membrane Transport Proteins Membrane Glycoproteins Membrane Transport Proteins Nerve Tissue Proteins Tritium (1R-(exo,exo))-3-(4-fluorophenyl)-8-methyl-8- azabicyclo(3.2.1)octane-2-carboxylic acid, methyl ester Sodium Cocaine Dopamine
Authors & Affiliations
4 authors, click to expand affiliations / ORCID
Reith M E
Department of Biomedical and Therapeutic Sciences, University of Illinois, College of Medicine, Peoria 61605, USA.
Xu C
Carroll F I
Chen N H
Article Info
Journal
Methods in enzymology
Abbr.
Methods Enzymol
ISSN
0076-6879
Published
1998-00-00
Pages
248-59
Language
English
Region
United States
NLM ID
0212271
Subset
IM
Grants
NIDA NIH HHS · DA 08379 · United States
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